تحضير وتشخيص و ودراسة النشاط البيولوجي والالتحام الجزيئي لبعض مشتقات السلفاميثوكسازول الجديدة.

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Al-Mudhafar M M J, Omeer T N-A, Abdul Hadi S L. Bis-Schiff Bases of Isatin Derivatives Synthesis, and their Biological Activities: A Review, Al Must J Pharm Sci. 2022; 22(1): 23-48. https://doi.org/10.32947/ajps.v22i1.827.

Li Q, Guan X, Wu P, Wang X, Zhou L, Tong Y, Ren R, at el. Early transmission dynamics in Wuhan, China, of novel coronavirus-infected pneumonia. N Engl. J Med. 2020; 382(13); 1199-1207. https://doi.org/10.1056/NEJMoa2001316.

Olyaei A, Sadeghpour M, Khalaj M. Mannich bases derived from lawsone and their metal complexes: synthetic strategies and biological properties, RSC Adv. 2020; 10: 30265-30281. https://doi.org/10.1039/D0RA05717G.

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Abdelgawad M A, Bukhari S NA, Musa A, Elmowafy M, Elkomy M H, Nayl A A, et. al. New Sulfamethoxazole Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors: Design, Synthesis, Cytotoxic Activity and Molecular Modeling. Pharmaceuticals. 2022; 15(9):1134. https://doi.org/10.3390/ph15091134.

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Elshihawy M M S, Abdel Aziz Y M , Elgawish MS, Elewa M, Elshihawy HA, Said MM. Pharmacophore modeling, 3D-QSAR, synthesis, and anti-lung cancer evaluation of novel thieno [2,3-d][1,2,3] triazines targeting EGFR. Arch Pharm. 2020; 353: 1900108. https://doi.org/10.1002/ardp.201900108.

Alkhaldi A A M, Al-Sanea M M, Nocentini A, Bonardi A, Lasheen D S, Elrazaz E Z, et al. 3-Methylthiazolo[3,2-a]benzimidazole-benzene sulfonamide conjugates as novel carbonic anhydrase inhibitors endowed with anticancer activity: design, synthesis, biological and molecular modeling studies. Eur J Med Chem. 2020; 207: 112745. https://doi.org/10.1016/j.ejmech.2020.112745.

Eldeeb A H, Abo-Ashour MF, Angeli A, Bonardi A, Lasheen D S, Elrazaz EZ, et al. Novel benzene sulfonamides aryl and aryl sulfone conjugates adopting tail/dual tail approaches: synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies. Eur J Med Chem. 2021; 221: 113486. https://doi.org/10.1016/j.ejmech.2021.113486.

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Sager G S, Salah A S, Mekky A H. Microwave Synthesis, Characterization of Some Novel Curcumin Compound and its Metal Complexes with Antimicrobial, Antioxidant Studies. Int J Med Pharm Res. 2020; 12(1): 429-448. https://doi.org/10.31838/ijpr/2020.12.01.200.

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Akili S, Hadda D B, Bitar Y, Balash A, Chehna MF. Design, Synthesis and Characterization of Novel Sulfonamides Derivatives as Anticancer Agent Targeting EGFR TK, and Development of New Methods of Synthesis by Microwave Irradiation. Int J Org Chem. 2021; 11(4): 119-123. https://doi.org/10.4236/ijoc.2021.114014.

Sangande F, Julianti E, Tjahjono D H. Ligand-Based Pharmacophore Modeling, Molecular Docking, and Molecular Dynamic Studies of Dual Tyrosine Kinase Inhibitor of EGFR. Int J Cell Sci Mol Biol. 2020; 21(20): 7779. https://doi.org/10.3390/ijms21207779.

Ibraheem I H, Mubder N S, Abdullah M A, Al-Neshmi H. Synthesis, characterization and bioactivity Study from azo –ligand derived frommethyl-2-amino benzoate with some metal ions. Baghdad Sci J. 2023; 20(1): 114-120. https://dx.doi.org/10.21123/bsj.2022.6584.

Rasheed A M, Al-Bayati S M M, Al-Hasani R A M, Shaker M A. Synthesizing Structure and Characterizing Bioactivities of Cr (III), La(III) and Ce(III)Complexes with Nitrogen ,Oxygen and Sulphur donor bidentate Schiff base ligands. Baghdad Sci. J. 2021;b18(4): 1547. https://doi.org/10.21123/bsj.2021.18.4(Suppl.).1545.

Abdul Kareem H M, Al-Tameemi M, Ibraheem I H, Sameer M. Surfactant Cloud Point Extraction as a Procedure of Preconcentrating for Metoclopramide Determination Using Spectro Analytical Technique. Baghdad Sci J . 2020; 17(1): 57-65. https://dx.doi.org/10.21123/bsj.2020.17.1.0057.

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